Table 3.
Free tissue : total plasma availability ratios
Treatment | AUCtissue i.m.: AUCplasma | AUCtissue s.c. : AUCplasma |
---|---|---|
Test A: DCF100C1 (1%) | 0.14 ± 0.24 (range 0.01–0.72; n = 8) | 0.10 ± 0.13 (range 0.01–0.47; n = 10) |
Test B: DCF100C2 (1%) | 0.12 ± 0.05 (range 0.03–0.21; n = 12) | 0.13 ± 0.12 (range 0.02–0.37; n = 11) |
Test C: DCF100C1 (2.5%) | 0.04 ± 0.04 (range 0.01–0.12; n = 11) | 0.05 ± 0.04 (range 0.01–0.12; n = 11) |
Test D: DCF100C2 (2.5%) | 0.85 ± 2.62 (range 0–8.76; n = 11) | 0.16 ± 0.22 (range 0.01–0.79; n = 11) |
Test E: Voltaren® Emulgel® | 0.62 ± 1.11 (range 0.02–3.36; n = 10) | 0.73 ± 1.33 (range 0.06–4.66; n = 11) |
Results are given as means ± SD (range).