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. 2011 Feb 8;54(5):1511–1528. doi: 10.1021/jm1015389

Table 3. Transcription/Translation (TnT) Assay Data.

compd E. colia MIC (μg/mL) TnT IC50 (μg/mL)
20f 0.125 0.76
20j 0.25 1.1
20k 0.25 0.93
21a 4 0.78
21b 8 0.36
21c 32 0.71
24i 8 0.58
24l 0.5 0.70
24c 4 5.3
24n 2 2.8
24o 32 3.4
tetracycline 2 2.0
tigecycline 0.125 0.47
a

ATCC 25922 is a tetracycline-susceptible strain.