Table 1.
No. | Ref. | Structure | Activity[a] (IC50) | Type of Inhibition |
---|---|---|---|---|
1 | [105] | >80% inhibition at 200 μM | No data | |
2 | [106] | 10 nM | Competitive with PAP | |
3 | [108] | 0.15 – 0.25 nM | Non-competitive | |
4 | [109] | 0.1 μM | Competitive | |
5 | [113] | 70 μM | Non-competitive | |
6 | [114] | 20 μM | Competitive | |
7 | [117] | 96 nM (Ki) | Competitive | |
8 | [99] | 50 μM | No data | |
9 | [99] | 30 μM | No data | |
10 | [119] | 30 μM | Specific, reversible | |
11 | [119] | 40 μM | Specific, irreversible |
Enzymes assayed: 1-4: EST; 5 : P-Selectin ; 6: GST; 7: β-AST-IV; 8: NodH; 9: GST-3; 10-11: TPST-2.