Fig. (4).

Compound Ranking. A) 9XGAL4UAS stable cell line was transiently transfected with pBIND-GR and then transferred to 384 well plates. One day after transfection, cells were induced with a serial dilution of agonists. B) Antagonists were serially diluted and added to cells in the presence of 100 nM Dex. C) 9XGAL4UAS stable cell line was transiently transfected with pBIND-ER. One day after transfection, cells were induced with a serial dilution of agonists. D) Antagonists were serially diluted and added to cells in the presence of 1.0 nM E2.