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. 2011 May 13;3:14. doi: 10.1186/1758-2946-3-14

Table 3.

Ranking of top-50 targets by numbers of compounds and documents.

Rank Approved
Symbol
Entrez Gene
ID
No of
compounds
No of
documents
1 F10 2159 42869 690

2 CNR1 1268 29658 578

3 KDR 3791 27661 350

4 MAPK14 1432 24568 309

5 DRD3 1814 23405 508

6 F2 2147 22853 768

7 HRH3 11255 22748 407

8 TACR1 6869 21908 626

9 MMP13 4322 20590 315

10 CNR2 1269 19712 464

11 MMP1 4312 17525 394

12 ADORA2A 135 17181 532

13 EGFR 1956 16581 445

14 SLC6A4 6532 16571 403

15 MMP9 4318 16537 344

16 HTR6 3362 16457 504

17 MMP2 4313 16405 310

18 HTR2C 3358 15945 475

19 CRHR1 1394 15550 222

20 MC4R 4160 15084 299

21 HTR2A 3356 14622 509

22 NPY5R 4889 14547 216

23 CCR3 1232 14136 114

24 OPRM1 4988 13394 466

25 DPP4 1803 13057 308

26 REN 5972 12894 438

27 CALCRL 10203 12615 137

28 CTSS 1520 12426 177

29 CHRM3 1131 12398 412

30 CCR2 729230 12208 160

31 DRD2 1813 12050 564

32 MET 4233 11745 118

33 ADORA1 134 11644 480

34 GSK3B 2932 11283 198

35 CCR5 1234 11179 197

36 CXCR2 3579 10851 183

37 SRC 6714 10838 282

38 MCHR1 2847 10821 209

39 EDNRA 1909 10769 260

40 NR3C1 2908 10687 199

41 EDNRB 1910 10601 239

42 HTR1A 3350 10015 627

43 OPRK1 4986 9690 375

44 TACR2 6865 9676 301

45 SLC6A2 6530 9671 272

46 ADORA3 140 9533 457

47 OPRD1 4985 9500 394

48 HSD11B1 3290 9334 151

49 ELANE 1991 9173 308

50 TRPV1 7442 8988 150