Table 1.
Percent growth inhibition obtained with the K562 cell line with compounds at 10 μM and IC50 values (μM) with the same cells.
| Com. | % inhibition | IC50 (μM) |
|---|---|---|
| 4 | 14.2 | >10 |
| 12a | 65.4 | 5.5 |
| 12b | 64.0 | 2.5 |
| 12c | 62.4 | 5.0 |
| 12d | 58.0 | 7.4 |
| 12e | 28.2 | >10 |
| 12f | 31.0 | >10 |
| 12g | 49.0 | 10 |
| 12h | 27.0 | >10 |
| 12i | 52.2 | 9.5 |
| 12j | 37.8 | >10 |
| 12k | 64.0 | 6.3 |
| 12l | 59.0 | 8.1 |
| 12m | 25.5 | >10 |
| 12n | 22.0 | >10 |
| 12o | 46.2 | >10 |
| 12p | 45.9 | >10 |
| 12q | 43.2 | >10 |
| 12r | 43.8 | >10 |
| 12s | 45.9 | >10 |
| 17t | 74.5 | 0.57 |
| 17u | 74.1 | 1.2 |
| 17v | 26.3 | >10 |
| 18 | 63.6 | 0.02 |