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. Author manuscript; available in PMC: 2012 Jun 27.
Published in final edited form as: J Chem Inf Model. 2011 May 25;51(6):1296–1306. doi: 10.1021/ci2000665

Table 3.

Some example complexes showing the relations between sp3 hybridized Carbon & sp2 hybridized Carbon VDW interaction, Zn chelation and pKd.

PDB Code VDW C3_C2 Zn Chelation pKd
1vkj −16.885 N/A 4.85
1a99 −12.084 N/A 5.70
1apb −15.76 N/A 5.82
1b58 −37.926 N/A 6.59
1lrh −28.539 N/A 6.82
1h2t −23.873 N/A 7.89
1fcy −60.245 N/A 8.52
1kdk −27.797 N/A 9.05
2fgu −45.694 N/A 9.18
1mrw −39.35 N/A 9.7
1df8 −42.823 N/A 9.92
1xpz −12.559 Y 7.08
1cny −15.87 Y 7.85
1ydb −3.7781 Y 8.24
1cim −12.885 Y 8.82
1cil −14.889 Y 9.43
1bnt −14.195 Y 9.89
1bnn −3.683 Y 10.00