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. Author manuscript; available in PMC: 2012 Jul 1.
Published in final edited form as: Nucl Med Biol. 2011 Mar 3;38(5):725–739. doi: 10.1016/j.nucmedbio.2011.01.002

Table 1.

In vitro Binding Data

Compound D2 D3 D4 D2:D3 Log P %IA D2 %IA D3
6 (WC-10) 34.4 ± 3.3 0.8 ± 0.1 896 ± 193 43 3.09 34 ± 3 19 ± 2
7 (WC-44) 54.7 ± 4.4 2.4 ± 0.4 804 ± 33 23 2.94 35 ± 1 96 ± 4
8 15.1 ± 1.7 0.65 ± 0.2 886 ± 101 23 3.75 66.3 ± 1 64.5 ± 8
9 27.7 ± 5.4 0.17 ± 0.01 246 ± 13.3 163 4.67 29.3 ± 7.3 34.4 ± 1.7