Syt4 and Syt7 are important for STD DA release, whereas Syt1 is essential for terminal DA release. A, STD DA release increases with time in culture. Extracellular [3H]DA levels were measured in DA neuron cultures in the presence of 0.5 mm Ca2+. B and C, down-regulation of Syt by siRNA. Cultured DA neurons were transfected at day 17 in culture using isoform-specific siRNA. The efficiency of transfection was 95%, and its effects on RNA (B) and protein (C) levels were assessed by semiquantitative RT-PCR and immunochemistry, respectively, at different days after transfection, as indicated. B, a representative gel of each Syt mRNA levels after siRNA transfection is shown. The presence of β-actin mRNA was evaluated to confirm the presence of mRNA and as a loading control. Note that Syt7 can be expressed as three different isoforms in mouse; DA neurons preferentially express Syt7a, the smallest one. C, summary graph presenting the Syt/TH ratio measured at different days after transfection, as indicated. The cells were fixed and subjected to immunochemistry, 10 images were captured from random fields at 40× (n = 6) and quantified with Metamorph software. D, effect of Syt mRNA down-regulation on STD [3H]DA release. Transfection was performed at day 17 in culture; their effects were evaluated 4 days later. STD [3H]DA release was evaluated in the presence of 0.5 mm extracellular Ca2+. E, summary graph showing that elevation of extracellular K+ in the presence of 0.5 mm extracellular Ca2+causes a substantial increase in [Ca2+]i levels in cultured DA neurons. F, after down-regulation of Syt4/7, high potassium depolarization fails to significantly elevate extracellular DA levels in the presence of 0.5 mm extracellular Ca2+. G, the effect of Syt mRNA down-regulation on total STD [3H]DA release (STD plus terminal) was also evaluated (in the presence of 2 mm Ca2+). Syt1 down-regulation caused a large decrease in DA levels, whereas Syt7 down-regulation caused a more modest decrease. scrm, cells transfected with scrambled siRNA; GFP, cells transfected with siRNA against GFP (heterologous control); Ctl, no siRNA used during transfection. The number of experiments for each condition is indicated inside the bars. *, p < 0.05 versus 21d (A) or versus Ctl (C–G). The error bars represent S.D.