Table 2.
entry | R | Yielda (9 : 10) | |
---|---|---|---|
| |||
1 | Me | 81 % (1.2 : 1) | |
2 | Et | 85 % (1.25 : 1) | |
3 | i-Pr | 90 % (1.8 : 1) | |
4 | n-Bu | 87 % (1.35 : 1) | |
5 | i-Bu | 93 % (1.4 : 1) | |
6 | t-Bu | 85 % (1.9 : 1) | |
7 | Bn | 87 % (1.5 : 1) |
Combined isolated yield
entry | R | Yielda (9 : 10) | |
---|---|---|---|
| |||
1 | Me | 81 % (1.2 : 1) | |
2 | Et | 85 % (1.25 : 1) | |
3 | i-Pr | 90 % (1.8 : 1) | |
4 | n-Bu | 87 % (1.35 : 1) | |
5 | i-Bu | 93 % (1.4 : 1) | |
6 | t-Bu | 85 % (1.9 : 1) | |
7 | Bn | 87 % (1.5 : 1) |
Combined isolated yield