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. 2011 Feb 23;63(3):255–259. doi: 10.1007/s12070-011-0151-8

Table 2.

Drugs causing tinnitus as a side effect

Drug category Class of drug Subclass of drug Examples
Anti infective Antibiotics Aminoglycosides Tobramycin, netilmicin, amikacin
Macrolides Clarithromycin, azithromycin
Quinolones Ciprofloxacin, ofloxacin, norfloxacin
Others Tetracyclines, vancomycin, teicioplanin, cotrimoxazole, cefpodoxime, linezolid
Antivirals Ganciclovir, zalcitabine,
Antifungals Amphotericin
Antimalarials Mefloquine, Quinine
Antituberculous Capreomycin
Analgesics diclofenac Non steroidal Aspirin, indomethacin, ibuprofen, diclofenac,
Anti-inflammatory Ketorolac, sulindac, naproxen, celecoxib
Anticancer drugs
Cardiac and vascular drugs
Cytotoxics Platinum compounds, Cisplatin, carboplatin
Vinca alkaloids Vindesine
Others Bexarotene, paclitaxel
Diuretics Loop diuretics Frusemide, torasemide
Potassium sparing diuretic Amiloride
Carbonic anhydrase inhibitor Acetazolamide
Beta blockers Metoprolol, timolol
Alpha blockers Prazocin
ACE inhibitor Ramipril, Enalapril, trandolapril
AT-II receptor Irbesartan
Antagonist
Anti arrhythmic Flecainide, quinidine, adenosine
Calcium channel blockers Diltiazem, nicardepine
Neurologic drugs Anticonvulsant Carbamazepine, fosphenytoin
Anti-depressant Tricyclics Imipramine, amitriptyline
SSRI Citalopram
Antimigraine 5HT-1 antagonist Almotriptan
Hypnotics Benzodiazepine (on withdrawal)
Others Immunosuppresant Tacrolimus
Antirheumatoid Hydroxychloroquine
Local anaesthetics Lignocaine
Hypoglycaemics Tolbutamide
Antihistamines Chlorpheniramine