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. Author manuscript; available in PMC: 2011 Oct 15.
Published in final edited form as: Org Lett. 2010 Oct 15;12(20):4438–4441. doi: 10.1021/ol101928m

Scheme 3.

Scheme 3

Cross-Coupling using Primary Amines

Reaction Conditions: ArX (0.5 mmol), amine (0.6 mmol), L5 (1 mol %), P5 (1 mol %), LiHMDS (1.2 mmol, 1 M in THF). Isolated yields are an average of at least two runs. aNo reaction when Pd(OAc)2 (1 mol %) used in place of P5. b Amine purified before use.