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CCR2 Antagonist MRL-677 Competition
| IC 50 or % inhibition | |
|---|---|
| Murine CCR2 | 1.8 ± 0.4 nM |
| Murine CCR5 | 418 ± 76 nM |
| Human CCR1 | 24% @ 10 μM |
| Human CCR3 | No inhibition @ 1 μM |
| Human CCR8 | No inhibition @ 1 μM |
| Human CXCR1 | 8% @ 10 μM |
| Human CXCR2 | 11% @ 1 μM |
| Human CXCR3 | 3% @ 1 μM |
