Table 1.
Voriconazole pharmacokinetic parameters in case patient and in healthy volunteers
Pharmacokinetic Parameter | Voriconazole 405 mg IV every 12h (case patient)* | Voriconazole 325 mg IV every 12h (case patient)+ | Voriconazole 4 mg/kg IV every 12h (healthy volunteers) (Purkins L et al., Antimicrob Agents Chemother 2002;46:2546–53) |
---|---|---|---|
AUC0–12 (ng · h/ml) | 77,790 | 104,245 | 29,467 |
Clearance (L/h) | 5.01 | 3.16 | ¶ |
Vd (L) | 221 | 101 | ¶ |
t1/2 (h) | 30 | 24 | 7.9 |
trough (mcg/ml) | 6.1 | 6.7 | 1.7 |
infusion time (1.75 h); collection time points from beginning of infusion (2.5, 5.6, 9.5, 11.5 h).
infusion time (1.5 h); collection time points from beginning of infusion (3.1, 6, 10.2, 12.2 h).
not reported.