Official websites use .gov
A
.gov website belongs to an official
government organization in the United States.
Secure .gov websites use HTTPS
A lock (
) or https:// means you've safely
connected to the .gov website. Share sensitive
information only on official, secure websites.
| entry | R | mGlu5 IC50 (nM) |
|---|---|---|
| 138 | 6-methylpyridin-2-yl | 65 |
| 261 | 4-methylthiazol-2-yl | 59 |
| 262 | 1-methyl-1H-pyrazol-3-yl | >10 000 |
| 263 | 4-cyclopropylthiazol-2-yl | 900 |
| 264 | phenyl | 5440 |
| 265 | 3-chlorophenyl | 45 |
| 266 | 3-methylphenyl | 122 |
| 267 | 3-chloro-2-fluorophenyl | 347 |
| 268 | 3-chloro-4-fluorophenyl | 377 |
