Table 3.
Fluorescence Polarization and Isothermal Titration Calorimetry Confirm the Flow Cytometry Data for Bcl-B
| Compound | FP Cy5-Bim log EC50 | FP F-Bim log EC50 | Flow F-Bim log EC50 | ITC compound log Kd |
|---|---|---|---|---|
| CID 650929 | −5.7 | −6.0 | −5.3 | −6.7 |
| CID 1243212 | −5.3 | −5.1 | −5.6 | −5.5 |
| CID 666339 | −6.0 | −6.0 | −5.7 | −5.6 |
| SID 85203040 | −6.0 | −6.0 | −5.7 | −5.6 |