Table 1.
Compound | IC50 (μM ± s.e.m.1) | logP | Water solubility (mM) |
---|---|---|---|
γ-Valerolactone | NI | 0.603 | 251 |
γ-Hexalactone | NI | 0.981 | 76 |
γ-Heptalactone | NI | 1.335 | 22 |
γ-Octalactone | 426 ± 438 | 1.668 | 7 |
γ-Nonalactone | 181 ± 18 | 1.985 | 2 |
γ-Decalactone | 43 ± 5 | 2.289 | 0.6 |
γ-Dodecalactone | 146 ± 25 | 2.861 | 0.057 |
Parthenolide | 105 ± 52 | 1.743 | 0.027 |
Costunolide | 233 ± 132 | 2.826 | 0.004 |
Santonin | 250 ± 312 | 1.598 | 0.285 |
β-Eudesmol | 3 ± 0.72 | 3.475 | 0.062 |
This table shows the IC50 values for decrease in planarian motility induced by the tested γ-lactones, as obtained from fitting the data in Figure 3 to equation 1. NI = No inhibition of movement.
Standard Error of the Mean.
From Pagán et al., (2008).