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. Author manuscript; available in PMC: 2012 Jan 1.
Published in final edited form as: Crit Rev Eukaryot Gene Expr. 2011;21(1):71–100. doi: 10.1615/critreveukargeneexpr.v21.i1.50

TABLE 3.

Clinical Trials Utilizing Drugs That Impact Autophagy”

Agent Target
Tamoxifen Estrogen receptor
Temozolomide DNA
γ-irradiation DNA
SAHA HDAC
Hyperthermia Unknown
Arsenic trioxide Mitochondria
Resveratrol Multiple
Rapamycin mTOR
Temsirolimus mTOR
Everolimus mTOR
2-deoxy-D-glucose Glycolysis
Endostatin Angiogenesis
Sorafenib TKI, VEGFR
Lonafarnib Farnesyltransferase