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. 2011 Jan 4;6(3):514–522. doi: 10.1002/cmdc.201000467

Table 1.

IC50 values of selected compounds against PI3Kα and PI3Kγ.

Compd IC50 [μm] Ratio
PI3Kα PI3Kγ α/γ
1 4.5 0.30 18
2 0.060 0.0080 7.5
3 0.050 0.040 1.3
4 0.25 0.10 2.5
5 0.45 0.12 3.8
6 50 >100 <0.50
7 1.9 1.0 1.9
8 7.3 27 0.30
9 4.4 9.3 0.50
10 2.7 4.9 0.60
11 0.069 0.042 1.6
12 0.15 0.12 1.2
13 2.7 0.25 11
14 11 1.5 7.1
15 9.4 3.1 3.1
16 86 4.0 22
17 22 1.4 16
19 0.0030 0.0013 2.2
20 8.3 0.62 13
40 3.0 0.41 7.3
41 11 1.4 7.9
42 0.14 0.060 2.3
43 8.7 >100 <0.087
44 9.0 >100 <0.090
45 0.40 0.20 2.0
46 0.10 0.025 4.0
47 0.80 1.0 0.80