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Group IVA PLA2 Inhibition by 1,3-Disubstituted Propan-2-ones In Vitro and in Cellular Assay
| Compound | IC50 (µM) | ||
|---|---|---|---|
| vesicle assay with the isolated enzyme |
cellular assay with human platelets stimulant A23187 |
cellular assay with human platelets stimulant TPA |
|
| 81a | 0.020 | 0.21 | 0.0078 |
| 81b | 0.0043 | 0.57 | 0.0009 |
