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. Author manuscript; available in PMC: 2012 Oct 12.
Published in final edited form as: Chem Rev. 2011 Sep 12;111(10):6130–6185. doi: 10.1021/cr200085w

Table 8.

Group IIA PLA2 Inhibition by Amides Derived from D-tyrosine

graphic file with name nihms324958t4.jpg
R IC50 (µM)
benzyl- 0.029
2-picolyl- 0.214
cyclopentylmethyl- 0.057
1-napthylmethyl- 0.019
2-napthylmethyl- 0.039
cinnamyl- 0.116
iso-butyl 0.170
n-heptyl 0.086
H 2.57