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. 2011 May-Jun;4(3):96–105.

Table 2.

Outcomes of studies of docetaxel and S-1 combinations

Author Regimen(s) No. of patients Study design, phase Tumor type Grade 3/4 neutropenia, % Other grade 3/4 AEs, n (%), and safety conclusion Median OS, months ORR, %
Kunisaki et al50 Docetaxel 20–45 mg/m2 days 1 and 15 + S-1 oral 80–120 mg/day, days 1–7 and days 15–21 21 I Advanced gastric adenocarcinoma n/a (DLT = neutropenia) n/a n/a 57.1
Park et al51 Docetaxel 35 mg/m2 days 1 and 8 + S-1 oral 40 mg/m2 bid days 1–14, q3w 52 II Metastatic gastric adenocarcinoma 29.4 Febrile neutropenia (19.6) 13.7 66.7
Sato et al52 Docetaxel 60 mg/m2 day 8 + S-1 oral 40 mg/m2 bid days 1–14, q3w 31 II Advanced or unresectable gastric adenocarcinoma 51.6 (grade 4: 32) Anorexia (29), nausea (26.6) n/a 87.1
Yamaguchi et al53 Docetaxel 40 mg/m2 day 1 + S-1 oral 40 mg/m2 bid days 1–14, q4w 46 II Advanced gastric adenocarcinoma 67 Leukopenia (41), anemia (22), anorexia (22), hyponatremia (17) 14.0 46
Yoshida et al54 Docetaxel 40 mg/m2 day 1 + S-1 oral 40 mg/m2 bid days 1–14, q3w 48 II Advanced or recurrent gastric adenocarcinoma 58.3 Febrile neutropenia (8.3), leukopenia (41.7), appetite loss (14.6) 14.3 56.3
Nakayama et al55 Docetaxel 40 mg/m2 + cisplatin 60–80 mg/m2 day 1 + S-1 40 mg/m2 bid days 1–14, q4w 14 I Advanced gastric adenocarcinoma n/a DLT: grade 3 diarrhea, febrile neutropenia, delayed resumption of treatment n/a n/a

Abbreviations: AE = adverse event; bid = twice daily; DLT = dose-limiting toxicity; n/a = not available; ORR = overall response rate; OS = overall survival; q3w = once every 3 weeks; q4w = once every 4 weeks.