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. Author manuscript; available in PMC: 2012 Nov 1.
Published in final edited form as: Clin Cancer Res. 2011 Aug 31;17(21):6944–6951. doi: 10.1158/1078-0432.CCR-11-0860

Table 2.

CYP2D6 metabolizer status based on genotype and drug inhibitor use.

CYP2D6
metabolizer
status
CYP2D6
genotype
CYP2D6 drug inhibitors
used
Weak
inhibitor
Potent
inhibitor
Ultra-rapid EM/UM,
UM/UM
no no
Extensive EM/EM no no
EM/UM,
UM/UM
yes no

Intermediate
EM/IM no no
EM/EM yes no
IM/IM no no
EM/PM no no
EM/IM yes no
EM/PM yes no
IM/IM yes no
PM/IM no no
Poor unknown no yes
any genotype no yes
PM/IM yes no
PM/PM no no
PM/PM unknown