Scheme 2.
PEGylation of 3′ amino-modified DNA A. PEGylation reaction of 3′ amino-modified DNA with N-hydroxysuccinimide PEG. B. PEGylation and decaging of DsRed targeting antisense DNA with the PhotoPEG reagent. C. Representative PAGE analysis of purified, PEGylated DNA. Lane 1: non-modified antisense agent (AA). Lane 2: 5 kDa PEGylated antisense agent (AA-5 kDa PEG). Lane 3: 20 kDa photocleavable PEGylated antisense agent (AA-5K PhotoPEG).
