. Author manuscript; available in PMC: 2012 Nov 15.

Published in final edited form as: Bioorg Med Chem Lett. 2011 Sep 20;21(22):6739–6745. doi: 10.1016/j.bmcl.2011.09.049

Table 6. S1P_1-5–Rs selectivity counter screen of compounds 24b, 24d, 24f (EC₅₀ nM).

^α

Data are reported as mean for n = 3 determinations.

^β

Percentage of response.

^χ

Percentage of inhibition at 25μM.

NA = not active at concentrations up to 25 μM.

Table 6. S1P1-5–Rs selectivity counter screen of compounds 24b, 24d, 24f (EC50 nM).