Table 4. IC50 or Ki values (μM) for inhibition of MMP-1, MMP-8, and MMP-13 by compounds 4, 20, and 24.
Target | Inhibitor | ||
---|---|---|---|
4 | 20 | 24 | |
MMP-1 (IC50) | >40 | >40 | >40 |
MMP-8 (IC50) | >40 | >40 | >40 |
MMP-13 (Ki) | 3.8 | 0.8 | 1.5 |
Target | Inhibitor | ||
---|---|---|---|
4 | 20 | 24 | |
MMP-1 (IC50) | >40 | >40 | >40 |
MMP-8 (IC50) | >40 | >40 | >40 |
MMP-13 (Ki) | 3.8 | 0.8 | 1.5 |