Table 2.
Average EC50 values for ER Ligands (M × 10−9)
| Hs578T-ERαLuc | Hs578T-ERβLuc | α/β | |
|---|---|---|---|
| E2 | 0.001 (0.0005) | 0.0065 (0.008) | 0.15 | 
| DPN | 8.5 (3) | 0.26 (0.02) | 33 | 
| PPT | 0.016 (0.001) | 26 (21) | 0.001 | 
| Liquiritigenin | 100 (40) | 28 (2) | 3.6 | 
Average EC50 values for ER Ligands (M × 10−9)
| Hs578T-ERαLuc | Hs578T-ERβLuc | α/β | |
|---|---|---|---|
| E2 | 0.001 (0.0005) | 0.0065 (0.008) | 0.15 | 
| DPN | 8.5 (3) | 0.26 (0.02) | 33 | 
| PPT | 0.016 (0.001) | 26 (21) | 0.001 | 
| Liquiritigenin | 100 (40) | 28 (2) | 3.6 |