Skip to main content
. Author manuscript; available in PMC: 2011 Dec 1.
Published in final edited form as: Exp Clin Psychopharmacol. 2008 Dec;16(6):446–457. doi: 10.1037/a0014196

Table 1. Monoamine Uptake Inhibition (IC50 nM).

Compound [3H]DA [3H]5HT Ratio 5HT/DA
Cocainea 310 260 0.8
RTI-112a 1.1 1.4 1.3
RTI-113a 3.0 229 76
RTI-177a 1.9 235 124
RTI-336b 12 522 44
GBR12909c 1.0 170 170
a

Data from Kuhar et al. (1999). Uptake values were determined using rat tissue.

b

Values supplied by NIDA under the Cocaine Treatment Discovery Program (CTDP) . Uptake values were determined using cloned hDAT and hSERT.

c

Data from Anderson (1989). Uptake values were determined using rat tissue.

HHS Vulnerability Disclosure