Table 2.

Inhibitory kinetics of vivapains and falcipains (Table has been taken from Na et al. 2004)

	kass (M−1 s−1)a
	Vivapain-2	Vivapain-3	Falcipain-2	Falcipain-3
E-64	2,31,000 ± 17,700	5,690 ± 588	14,200 ± 475	5,870 ± 428
Z-Phe-Arg-FMK	47,900 ± 5,090	3,680 ± 218	2,41,000 ± 20,100	60,200 ± 6,740
Mu-Phe-hPhe-FMK	61,700 ± 6,180	540 ± 60	2,15,000 ± 5,760	5,26,000 ± 59,300
Mu-Leu-hPhe-FMK	4,50,000 ± 16,800	79,200 ± 6,490	9,24,000 ± 26,200	58,50,000 ± 15,800
Mu-Phe-hPhe-VSph	267 ± 14	NAb	4,890 ± 231	2,060 ± 41
Mu-Leu- hPhe-VSph	88,200 ± 470	4,970 ± 370	1,02,000 ± 2,530	22,000 ± 1,420
Nmetpip-Phe-hPhe-VSPh	96 ± 5	15 ± 004	1,230 ± 136	1,900 ± 43
Nmetpip-Leu-hPhe-VSPh	53,600 ± 6,450	2,130 ± 158	26,300 ± 3,700	11,900 ± 762

Mu morpholine urea, hPhe homophenylalanine, NmetpipN-methylpiperazine urea, VSPh phenylvinylsulphone

^aGeometric mean ± SEM

^bNo appreciable activity