TABLE 1.
Antagonist and Concentration | EROD Activity (Percentage of 10 nM TCDD) |
||
---|---|---|---|
HaCaT | HepG2 | T84 | |
% | % | % | |
CH223191 | |||
1 μM | 33 ± 6 | 58 ± 16 | 30 ± 8 |
CHD-5 | |||
1 μM | 27 ± 6 | 58 ± 13 | 29 ± 8 |
10 μM | 21 ± 11 | 28 ± 9 | 28 ± 9 |
CHD-7 | |||
1 μM | 104 ± 10*† | 82 ± 9‡ | 94 ± 9*† |
10 μM | 96 ± 4 | 98 ± 16‡ | 68 ± 3 |
CHD-8 | |||
1 μM | 113 ± 4*† | 68 ± 7 | 103 + 9*† |
10 μM | 109 ± 9 | 79 ± 7 | 87 ± 2*† |
CHD-11 | |||
1 μM | 36 ± 10 | 33 ± 10 | 32 ± 7 |
10 μM | 23 ± 3 | 29 ± 9 | 28 ± 9 |
CHD-12 | |||
1 μM | 29 ± 7 | 34 + 8 | 31 ± 8 |
10 μM | 21 ± 2 | 29 + 9 | 24 ± 10 |
Statistically different (P < 0.05) from CH223191.
Statistically different (P < 0.05) from CHD-5, CHD-11, and CHD-12 at the corresponding concentrations.
Statistically different (P < 0.05) from CHD-11 and CHD-12 at the corresponding concentrations.