TABLE 1.

IC₅₀ values and % inhibition from competition binding to apoB-100 with [¹²⁵I]T₁AM

Compounds	IC50	% of inhibition at 1 μm concentration of inhibitorsa
	nm
T1AM	5	91
3′-T1AM	259	48
T0AM	268	54
3,5-T2AM	209	72
3,3′-T2AM	570	62
T3AM	224	62
rT3AM	865	37
T4AM	3834	32
T0		14
T1		24
3,5-T2	738	56
3,3′-T2	776	54
T3	479	53
rT3	818	34
T4	1518	21
Tyramine		3
Serotonin		3

^a Percent inhibition at 1 μm concentration of inhibitors was determined in a separate experiment.