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. Author manuscript; available in PMC: 2013 Jan 12.
Published in final edited form as: J Med Chem. 2011 Dec 28;55(1):342–356. doi: 10.1021/jm201229j

Figure 2.

Figure 2

Effects of compound 4m on inhibtion of cAMP production induced by full agonist 1a at the hA3AR expressed in CHO cells (A). The data was transformed to a linear Schild plot (B) indicating competitive antagonism with a KB value of 23.9 nM.