Accumulation in transporter transfected cells (pmol/mg) | Accumulation in parental cells (1) (pmol/mg) | Highest Fold Activation | |||||||
Transporter | 2 min | 20 min | 2 min | 20 min | |||||
100 µM | 300 µM | 100 µM | 300 µM | 100 µM | 300 µM | 100 µM | 300 µM | ||
PEPT1 | 1073 | 2290 | 1087 | 1682 | 969 | 2389 | 981 | 1614 | 1.1 (100µM, 20 min) |
PEPT2 | 937 | 1871 | 897 | 1759 | 965 | 2011 | 1219 | 2056 | 0.97 (100µM, 20 min) |
50 µM | 100 µM | 50 µM | 100 µM | 50 µM | 100 µM | 50 µM | 100 µM | ||
OCT1 | 3818 | 5878 | 5540 | 9190 | 3894 | 6337 | 5672 | 9576 | Not observed |
OCT2 | 8492 | 15071 | 8866 | 15495 | 5660 | 8000 | 5790 | 8459 | 1.88 (100µM, 2 min) |
100 µM | 300 µM | 100 µM | 300 µM | 100 µM | 300 µM | 100 µM | 300 µM | ||
OATP2B1 | 11317 | 18296 | 20820 | 45866 | 6409 | 10891 | 10889 | 21496 | 2.1 (300 µM, 20 min) |