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. 2012 Feb 15;3:RRN1291. Originally published 2011 Dec 15. [Version 2] doi: 10.1371/currents.RRN1291
  Accumulation in transporter transfected cells (pmol/mg) Accumulation in parental cells (1) (pmol/mg) Highest Fold Activation
Transporter 2 min 20 min 2 min 20 min
  100 µM 300 µM 100 µM 300 µM 100 µM 300 µM 100 µM 300 µM
PEPT1 1073 2290 1087 1682 969 2389 981 1614 1.1
(100µM, 20 min)
PEPT2 937 1871 897 1759 965 2011 1219 2056 0.97
(100µM, 20 min)
  50 µM 100 µM 50 µM 100 µM 50 µM 100 µM 50 µM 100 µM  
OCT1 3818 5878 5540 9190 3894 6337 5672 9576 Not observed
OCT2 8492 15071 8866 15495 5660 8000 5790 8459 1.88
(100µM, 2 min)
  100 µM 300 µM 100 µM 300 µM 100 µM 300 µM 100 µM 300 µM  
OATP2B1 11317 18296 20820 45866 6409 10891 10889 21496 2.1
(300 µM, 20 min)