| Transporter | Incubation time (min) | Probe substrate (concentration) |
Reference inhibitor
(concentration) |
| human OATP2B1 | 15 | E3S (1 μM) | Fluvastatin (10 μM) |
| human OAT3 | 5 | E3S (0.3 µM) | Probenecid (500 µM) |
| human OCT1 | 10 | TEA (3.6 μM) | Verapamil (100 μM) |
| human OCT2 | 10 | Metformin (2 µM) | Verapamil (100 µM) |
| human PEPT1 | 10 | Gly-Sar (1.8 μM) | Tyr-Phe (200 μM) |
| human PEPT2 | 10 | Gly-Sar (1.8 μM) | Cefadroxil (200 μM) |
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