Skip to main content
. 2011 Oct 5;2(12):877–881. doi: 10.1021/ml2001246

Table 2. IC50 Data for Inhibition of Key Cytochrome P450 Isozymes.

CYP450 isozyme substrate/stock solution conc (μM) protein (mg/mL) incubation (min) IC50 data (μM)
CYP3A4 testosterone (50 mM) 100 0.3 30 >200
CYP3A4 triazolam (50 mM) 200 0.4 30 >200
CYP2D6 dextromethorphan (50 mM) 200 2.0 60 >200
CYP2C8 amodiaquine (5 mM) 200 0.4 30 >65