Table 2.
Evaluation of drug likeness properties.
| Compounds | MW <500 | C log P <5 | Number of O and N <10 | Number of OH and NH <5 | N rotatable bonds <10 | N-violations ≯1 |
|---|---|---|---|---|---|---|
| 1a | 306.32 | 1.44 | 5 | 0 | 3 | 0 |
| 1g | 340.76 | 1.97 | 5 | 0 | 3 | 0 |
| 1h | 375.20 | 2.45 | 5 | 0 | 3 | 0 |
| 1l | 351.31 | 1.35 | 8 | 0 | 4 | 0 |