Table 11.
Cross-coupling reactions of heteroaryl chlorides and heteroaryl secondary aminesa
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ArCl (1.0 mmol), amine (1.2 mmol).
amine (2 mmol).
0.5 mmol scale.
Cs2CO3/t-BuOH.
3% reduction of ArCl.
4% reduction of ArCl.
45 °C.
45 °C, SPhos.
Cross-coupling reactions of heteroaryl chlorides and heteroaryl secondary aminesa
![]() |
ArCl (1.0 mmol), amine (1.2 mmol).
amine (2 mmol).
0.5 mmol scale.
Cs2CO3/t-BuOH.
3% reduction of ArCl.
4% reduction of ArCl.
45 °C.
45 °C, SPhos.