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. Author manuscript; available in PMC: 2012 Dec 22.
Published in final edited form as: J Med Chem. 2011 Nov 23;54(24):8471–8489. doi: 10.1021/jm201018g

Table 7.

Structures and activities of analogues 26a – 26ja

graphic file with name nihms340444u7.jpg
Compound R1 IC50 (μM) Compound R1 IC50 (μM)
26a graphic file with name nihms340444t30.jpg 1.3 26f graphic file with name nihms340444t31.jpg 6.2
26b graphic file with name nihms340444t12.jpg 0.9 26g graphic file with name nihms340444t25.jpg 6.6
26c graphic file with name nihms340444t32.jpg >25 26h graphic file with name nihms340444t33.jpg 0.7
26d graphic file with name nihms340444t34.jpg 0.6 26i graphic file with name nihms340444t35.jpg 0.25
26e graphic file with name nihms340444t29.jpg 0.8 26j graphic file with name nihms340444t36.jpg 5.7
a

Results were from single runs