Table 3.
Compounds examined in the secondary screen
Code | MLS # | Vendor | Vendor Cat # | IC50 (μM) |
---|---|---|---|---|
A | MLS000075845 | Asinex | BAS 08769335 | 13.3 |
B | MLS000035239 | Asinex | ASN 05830127 | 4.7 |
C | MLS000075919 | Asinex | BAS 07869980 | 2.1 |
D | MLS000035419 | Asinex | BAS 06754276 | 9.9 |
E | MLS000073086 | Asinex | BAS 04834866 | 2.5 |
F | MLS000068249 | Asinex | ASN 04363458 | 9.4 |
G | MLS000027771 | Asinex | BAS 09533241 | 15.3 |
H | MLS000031372 | Asinex | BAS 00506290 | 10.9 |
I | MLS000071970 | Asinex | BAS 00506281 | 24.7 |
N | MLS000051260 | ChemBridge | 7925560 | 6.8 |
P | MLS000111675 | ChemBridge | 6370266 | >40 |
J | MLS000105542 | ChemBridge | 5161874 | 12.6 |
O | MLS000108799 | ChemBridge | 5927508 | 7.7 |
M | MLS000049833 | ChemBridge | 7894782 | 16.5 |
L | MLS000096979 | ChemBridge | 7685300 | >40 |
R | MLS000062315 | ChemBridge | 6624994 | 3.6 |
Q | MLS000062185 | ChemBridge | 6512965 | 3.4 |
K | MLS000104229 | ChemBridge | 5215570 | 10.3 |
C′ | MLS000047713 | ChemDiv | 2324-0448 | 12.0 |
B′ | MLS000092741 | ChemDiv | C656-0067 | 23.3 |
W | MLS000109390 | Deltagen | 4065-0146 | 4.3 |
V | MLS000073581 | Deltagen | K408-0544 | 4.8 |
X | MLS000057191 | EnAmine | T5347014 | 8.4 |
Y | MLS000057778 | EnAmine | T0511-0376 | 13.3 |
Z | MLS000055414 | EnAmine | T0507-2864 | 8.1 |
U | MLS000069631 | Sigma | C1386 | 10.3 |
T | MLS000043319 | ChemBridge | 7461374 | 0.9 |
S | MLS000106248 | ChemBridge | 5344221 | 1.7 |
A′ | MLS000045466 | ChemDiv | C505-0274 | 3.5 |
D′ | MLS000041467 | ChemDiv | 6917-0116 | 4.0 |