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. Author manuscript; available in PMC: 2012 Mar 11.
Published in final edited form as: Bioorg Med Chem. 2008 Mar 6;17(3):990–1005. doi: 10.1016/j.bmc.2008.03.004

Table 3.

Compounds examined in the secondary screen

Code MLS # Vendor Vendor Cat # IC50 (μM)
A MLS000075845 Asinex BAS 08769335 13.3
B MLS000035239 Asinex ASN 05830127 4.7
C MLS000075919 Asinex BAS 07869980 2.1
D MLS000035419 Asinex BAS 06754276 9.9
E MLS000073086 Asinex BAS 04834866 2.5
F MLS000068249 Asinex ASN 04363458 9.4
G MLS000027771 Asinex BAS 09533241 15.3
H MLS000031372 Asinex BAS 00506290 10.9
I MLS000071970 Asinex BAS 00506281 24.7
N MLS000051260 ChemBridge 7925560 6.8
P MLS000111675 ChemBridge 6370266 >40
J MLS000105542 ChemBridge 5161874 12.6
O MLS000108799 ChemBridge 5927508 7.7
M MLS000049833 ChemBridge 7894782 16.5
L MLS000096979 ChemBridge 7685300 >40
R MLS000062315 ChemBridge 6624994 3.6
Q MLS000062185 ChemBridge 6512965 3.4
K MLS000104229 ChemBridge 5215570 10.3
C′ MLS000047713 ChemDiv 2324-0448 12.0
B′ MLS000092741 ChemDiv C656-0067 23.3
W MLS000109390 Deltagen 4065-0146 4.3
V MLS000073581 Deltagen K408-0544 4.8
X MLS000057191 EnAmine T5347014 8.4
Y MLS000057778 EnAmine T0511-0376 13.3
Z MLS000055414 EnAmine T0507-2864 8.1
U MLS000069631 Sigma C1386 10.3
T MLS000043319 ChemBridge 7461374 0.9
S MLS000106248 ChemBridge 5344221 1.7
A′ MLS000045466 ChemDiv C505-0274 3.5
D′ MLS000041467 ChemDiv 6917-0116 4.0