(A,B) PITs inhibit ARF6-induced cell migration. SUM159 cells were transfected with ARF6. Scratch wound was generated in cell monolayer, followed by treatment with PITs (50 μM) for 8 hr. The width of wounded cell monolayers was measured in five random fields and expressed as % of original width (A). The wound width ratio (PITs treated groups/DMSO control group) was calculated (B).
(C) Overexpression of ARF6-Q67L attenuates inhibition of cell migration led by PIT-1. SUM159 cells were transfected with ARF6-Q67L. Scratch wound was generated in cell monolayer, followed by treatment with compounds for 8 hr. The width of wounded cell monolayer was measured in five random fields, and the inhibition was calculated.
(D,E) PITs inhibit GRP1/ARNO-induced cell migration. SUM159 cells were transfected with full length GRP1 or ARNO. Scratch wound was generated in cell monolayer, followed by treatment with PITs (50 μM) for 8 hr. The width of wounded cell monolayers was measured in five random fields and expressed as % of original width (D). The wound width ratio (PITs treated groups/DMSO control group) was calculated (E).
(F) Overexpression of EFA6 attenuates inhibition of cell migration by PIT-1. SUM159 cells were transfected with EFA6. Scratch wound was generated in cell monolayer, followed by treatment with compounds for 8 hr. The width of wounded cell monolayer was measured in five random fields, and the inhibition was calculated.
*P<0.05, **P<0.01 compared with empty vector group.