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. 2012 Jan 10;119(9):1992–2002. doi: 10.1182/blood-2011-06-354647

Table 1.

Small molecules used in screening

17-AAG CHIR258 JAK1i Nilotinib SB-43152
8 Azaguanine CHIR265 JAK3i P38i SB203580
ABT-864 CI-1033 JNK2i Pan-JAKi Sorafenib
Adiphenine CP-690550 JNKIIi PD153035 SRCi
AG490 CYC-202 KN92 PD325901 Staurosporine
AKTIV Dasatinib KN93 PD98059 STO609
AKTX EGFRi Lapatinib PI-103 Sunitinib
AMPK Erlotinib LSD1 Piperine SYKi
Anisomycin Estradiol LY294002 PKC412 Thapsigargin
AZD-1152 Gefitinib LY333531 PP2 Trichostatin A
Azithromycin Go6976 MEK1/2 Proguanil Tunicamycin
BAY-11 GW-786034 Menadione PTK787 Vorinostat
BIRB-796 H-89 MLN-8054 R1881 VX-680
Boldine Harmane MLN518 Resveratrol Zardaverine
cAMP Imatinib QNZ SB-202190 ZD-6474

For each molecule, at least 3 doses were tested. Cell viability was quantified using the 3-(4,5-dimethylthiazol-2-yl)-5-(3-carboxymethoxyphenyl)-2-(4-sulfophenyl)-2H-tetrazolium assay.