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. 2009 Jul;1(2):15–25.

Table 1.

Certain marine natural compounds are potential anticancer drugs

Compound Biological source Chemical nature Action mechanism Company Status
Bryostatin-1 (7) Bryozoan Poliketide Inhibitor of protein kinase GPC Biotech Phase 2 clinical trials
Dolastatin-10 (8) Mollusc Peptide Inhibitor of microtubeles formation NCI-Knoll Phase 2 clinical trials of its derivative TZT-1027
HTI286 (9) Sponge Tripeptide Inhibitor of microtubeles formation Novartis Continuation of clinical trials
Discodermalide (10) Sponge Poliketide Inhibitor of microtubeles formation Novartis Phase 2 clinical trials
Cryptophycin (11) Cyanobacterium Cyclic depsipeptide Inhibitor of microtubeles formation Eli Lilly Taken out from phase 2 clinical trials
Aplidin (12) Ascidian Cyclic depsipeptide Causes oxidative stress in cells PharmaMar Phase 2 clinical trials
Eribulin mesylate (13) Sponge Polyether derivative Inhibitor of microtubeles formation Esai Company Phase 3 clinical trials
Squalamine (14) Shark Steroid Inhibitor of angiogenesis Genaera Taken out from phase 2 clinical trials
Kohalalide F (15) Mollusc Cyclic depsipeptide Active on lysosomal level PharmaMar Phase 2 clinical trials
Salinosporamide A (16) Marine bacterium Lactam-lactone derivative Proteosome inhibitor Nereus Phase 2 clinical trials