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. 2012 Apr 19;2012:212178. doi: 10.1100/2012/212178

Table 3.

Inhibitors of CYP3A4.

(1) Antihypertensive medications
 Dihydralazine
 Diltiazem
 Verapamil
(2) Antidepressant and anxiolytic medications
 Fluoxetine
 Midazolam
(3) Antimicrobial medications
 Macrolides
 Clarithromycin
 Erythromycin
 Isoniazid
 HIV agents
(4) Endocrine medications
 Contraceptives
 Ethinylestradiol
 Antiprogesterone agent
 Estrogen receptor modulators
 Tamoxifen
(5) Food and herbal constituents
 Bergamottin (grapefruit juice)
 Glabridin (licorice)