Table 3.
Inhibitors of CYP3A4.
| (1) Antihypertensive medications |
| Dihydralazine |
| Diltiazem |
| Verapamil |
| (2) Antidepressant and anxiolytic medications |
| Fluoxetine |
| Midazolam |
| (3) Antimicrobial medications |
| Macrolides |
| Clarithromycin |
| Erythromycin |
| Isoniazid |
| HIV agents |
| (4) Endocrine medications |
| Contraceptives |
| Ethinylestradiol |
| Antiprogesterone agent |
| Estrogen receptor modulators |
| Tamoxifen |
| (5) Food and herbal constituents |
| Bergamottin (grapefruit juice) |
| Glabridin (licorice) |