Table 3.
| |||||
---|---|---|---|---|---|
entry | R | product | time (h) | C-4:C-6a | yield (%)b |
1 | -CH2CH3 | 6a | 8 | 90:10 | 53 |
2 | -CH3 | 6b | 10 | 93:7 | 44 |
3 | -CH2Ph | 6c | 10 | >95:5 | 45 |
Ratio determined by 1H NMR spectroscopy of the crude reaction mixture. All reactions were run at a concentration of 0.15 M with respect to 2.
Isolated yield of the C-4 regioisomer