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. Author manuscript; available in PMC: 2013 Jun 15.
Published in final edited form as: Bioorg Med Chem Lett. 2012 Apr 30;22(12):3921–3925. doi: 10.1016/j.bmcl.2012.04.112

Figure 3.

Figure 3

Library optimization strategy for VU0092273 (3) to improve mGlu3 NAM activity while simultaneously eliminating mGlu5 PAM activity.