. 2010 Dec 10;2(2):60–74. doi: 10.1021/cn1001039

Table 10. Functional Characterization (K_B) of Antagonists 9.1 and 9.2 in a TEVC Oocyte Assay at Cloned Non-Desensitizing Homomeric Subtypes GluK1-3^a.

cmpd	GluA1/2	GluK1	GluK2	GluK3
9.1^c	−^f	11.4	>300	273
9.2 ((S)-ATPO)^d	3.6^b	24^b	>300^e	−^f

All values in [μM].

Inhibition of KA-induced responses in Xenopus oocytes (K_i).

From ref (102).

From ref (104)

From ref (107).

Not tested.

Table 10. Functional Characterization (KB) of Antagonists 9.1 and 9.2 in a TEVC Oocyte Assay at Cloned Non-Desensitizing Homomeric Subtypes GluK1-3a.