Table 7.
Frequency of micronuclei in the bone marrow of mice treated with phospho-ibuprofen
| Treatment | Sex | Dose (mg/kg) | Time in Hours | n | PCE/RBC (%) Mean ± S.E. | PCE with MN (%) Mean ± S.E. |
|---|---|---|---|---|---|---|
| Control | Male | 0 | 24 | 5 | 47.46 ± 3.03 | 0.15 ± 0.03 |
| Phospho-Ibuprofen | Male | 500 | 24 | 5 | 52.60 ± 2.42 | 0.10 ± 0.03 |
| Phospho-Ibuprofen | Male | 1000 | 24 | 5 | 49.02 ± 2.63 | 0.10 ± 0.02 |
| Phospho-Ibuprofen | Male | 2000A | 24 | 4 | 49.94 ± 2.33 | 0.21 ± 0.06 |
| Urethane | Male | 300 | 24 | 5 | 51.10 ± 2.39 | 2.17 ± 0.26** |
| Control | Female | 0 | 24 | 5 | 48.54 ± 1.64 | 0.12 ± 0.04 |
| Phospho-Ibuprofen | Female | 500 | 24 | 5 | 44.84 ± 1.74 | 0.13 ± 0.05 |
| Phospho-Ibuprofen | Female | 1000 | 24 | 5 | 50.10 ± 0.53 | 0.15 ± 0.02 |
| Phospho-Ibuprofen | Female | 2000 | 24 | 5 | 53.44 ± 4.86 | 0.20 ± 0.02 |
| Control | Male | 0 | 48 | 5 | 48.33 ± 1.57 | 0.14 ± 0.02 |
| Phospho-Ibuprofen | Male | 500 | 48 | 5 | 50.95 ± 2.77 | 0.04 ± 0.02 |
| Phospho-Ibuprofen | Male | 1000 | 48 | 5 | 52.31 ± 2.86 | 0.12 ± 0.03 |
| Phospho-Ibuprofen | Male | 2000 | 48 | 5 | 46.94 ± 2.55 | 0.18 ± 0.01 |
| Control | Female | 0 | 48 | 5 | 49.61 ± 2.76 | 0.11 ± 0.04 |
| Phospho-Ibuprofen | Female | 500 | 48 | 5 | 51.92 ± 3.84 | 0.18 ± 0.05 |
| Phospho-Ibuprofen | Female | 1000 | 48 | 5 | 46.36 ± 1.53 | 0.11 ± 0.03 |
| Phospho-Ibuprofen | Female | 2000 | 48 | 5 | 46.95 ± 0.91 | 0.08 ± 0.03 |
= One male mouse in this group found dead before necropsy; n = Number of surviving animals; PCE = Polychromatic erythrocytes; RBC= Red blood cells; MN = Micronuclei; Control = PEG 400;
= p < 0.05 by test for binomial proportions for test article;
= p < 0.01 by test for binomial proportions for positive control