Table 1.
Compound | r1 Tris Buffer | r1 fibrin | % Increase | Ki DD(E) (μM) |
---|---|---|---|---|
PepN-Gd4-NPep | 18.2 | 23.1 | 27 | 1.1 |
Gd4-NPep | 15.5 | 20.7 | 33 | 4.7 |
NPep-Gd4 | NR | NR | NR | 9.1 |
Gd2A-NPep-Gd2A | NR | NR | NR | 12.0 |
Gd2B-NPep-Gd2B | 13.0 | 18.0 | 37 | 4.7 |
Gd2-Gly2-NPep-Gd2 | 12.4 | 17.8 | 37 | 4.0 |
Gd2-T-NPep-Gd2 | 13.3 | 28.0 | 114 | 3.5 |