Table 1.
The examined data sets and their data types.
Set | Compounds | Congeneric? | Data type (N) | Reference |
---|---|---|---|---|
Avdeef | FDA drugs | No | PAMPA (11) | 66 |
Caco-2 (11) | ||||
Balamine | FDA drugs | No | PAMPA (22) | 67 |
Caco-2 (21) | ||||
%Abs (22) | ||||
Bermejo | Fluoroquinolones | Yes | PAMPA (16) | 68 |
Caco2 (14) | ||||
Perfusion assay (16) | ||||
Di | FDA drugs | No | PAMPA (27) | 69 |
Fujikawa | FDA drugs & small chemicals | No | PAMPA (70) | 70 |
Caco-2 (29) | ||||
Goodwin | Peptidomimetics | Yes | Caco-2 (12) | 71 |
Irvine | FDA drugs | No | Caco-2 (50) | 72 |
MDCK (51) | ||||
%Abs (53) | ||||
Li | Peptidomimetics | Yes | PAMPA (25) | 73 |
Caco-2 (25) | ||||
Whitlock | 1-(2-Phenoxyphenyl) methanamines | Yes | PAMPA (8) | 74 |