Table 1.
Entry | Alkaloids | Natural ([α]10D) | Synthetic ([α]24D)a |
---|---|---|---|
1 | Trigonoliimine A | +13.3 (c 0.3, CHCl3) | −294 (c 0.24, CHCl3, 94% ee) |
2 | Trigonoliimine B | +5.0 (c 0.5, CHCl3) | −352 (c 0.32, CHCl3, 95% ee) |
3 | Trigonoliimine C | −4.8 (c 0.45, CHCl3) | −147 (c 0.12, CHCl3, 96% ee) |
% ee of the key precursor for the corresponding synthetic trigonoliimine.